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G-Protein antagonist peptide TFA competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors
the activity of CZ415 against the human cardiac ion channel hERG is assessed in a whole-cell patch-clamp assay in HEK293 cells resulting in an IC50 of 48 μM
ML314 displays good brain penetration in rodents
which contributes to the current understanding of the functional association between PPZ and PKM2(The human M2 isoform of pyruvate kinase)[2]
and inhibits colony formation of hepatocarcinoma cells expressing FGFR1/2 and AXL
TC OT 39 Catalog No.:M23225-C G-Protein antagonist peptide TFA competitivelyProduct information CAS Number: 479232 57 0 Molecular Weight: 600. 78 Formula: C32H40N8O2S Chemical Name: (Z,2S) 2 (4 methyl 1,4 diazepane 1 carbothioyl) N [(2 methyl 4 {4 methyl 2,4,5,9 tetraazatricyclo[8. 4. 0. 0,]tetradeca 1(14),3(7),5,10,12 pentaene 9 carbonyl}phenyl)methyl]pyrrolidine 1 carboximidic acid Smiles: CC1=CC(=CC=C1C N=C(\O) N1CCC[C@H]1C(=S)N1CCCN(C)CC1)C(=O)N1CC2C=NN(C)C=2NC2=CC=CC=C12 InChiKey: KSNHHKZYKYNBEI NDEPHWFRSA N InChi:
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